Number of items: 46.
2023
Morgan, D. C., McDougall, L., Knuhtsen, A. and Jamieson, A.
(2023)
Development of bifunctional, Raman active diyne‐girder stapled α‐helical peptides.
Chemistry: A European Journal,
(doi: 10.1002/chem.202300855)
(PMID:37130830)
(Early Online Publication)
2022
Archibald, L. J., Brown, E. A., Millard, C. J., Watson, P. J., Robertson, N. S., Wang, S., Schwabe, J. W. R. and Jamieson, A. G.
(2022)
Hydroxamic acid-modified peptide library provides insights into the molecular basis for the substrate selectivity of HDAC corepressor complexes.
ACS Chemical Biology, 17(9),
pp. 2572-2582.
(doi: 10.1021/acschembio.2c00510)
(PMID:35973051)
(PMCID:PMC9488896)
Mahindra, A. et al.
(2022)
Investigating the structure–activity relationship of 1,2,4-triazine G-protein-coupled receptor 84 (GPR84) antagonists.
Journal of Medicinal Chemistry, 65(16),
pp. 11270-11290.
(doi: 10.1021/acs.jmedchem.2c00804)
(PMID:35948061)
(PMCID:PMC9421653)
Yelland, T. et al.
(2022)
Stabilization of the RAS:PDE6D complex is a novel strategy to inhibit RAS signaling.
Journal of Medicinal Chemistry, 65(3),
pp. 1898-1914.
(doi: 10.1021/acs.jmedchem.1c01265)
(PMID:35104933)
(PMCID:PMC8842248)
2021
Mahindra, A. et al.
(2021)
Peptides derived from the SARS-CoV-2 receptor binding motif bind to ACE2 but do not block ACE2-mediated host cell entry or pro-inflammatory cytokine induction.
PLoS ONE, 16(11),
e0260283.
(doi: 10.1371/journal.pone.0260283)
(PMID:34793553)
(PMCID:PMC8601423)
Morgan, D. C. et al.
(2021)
Stapled ACE2 peptidomimetics designed to target the SARS-CoV-2 spike protein do not prevent virus internalisation.
Peptide Science, 113(4),
e24217.
(doi: 10.1002/pep2.24217)
(PMID:33615115)
(PMCID:PMC7883042)
Knuhtsen, A., Whiting, R., McWhinnie, F. S., Whitmore, C., Smith, B. O. , Green, A. C., Timperley, C. M., Kinnear, K. I. and Jamieson, A. G.
(2021)
μ-conotoxin KIIIA peptidomimetics that block human voltage-gated sodium channels.
Peptide Science, 113(1),
e24203.
(doi: 10.1002/pep2.24203)
2020
Mahindra, A., Janha, O., Mapesa, K., Sanchez Azqueta, A., Alam, M. M. , Amambua-Ngwa, A., Nwakanma, D. C., Tobin, A. B. and Jamieson, A. G.
(2020)
Development of potent PfCLK3 inhibitors based on TCMDC-135051 as a new class of antimalarials.
Journal of Medicinal Chemistry, 63(17),
pp. 9300-9315.
(doi: 10.1021/acs.jmedchem.0c00451)
(PMID:32787140)
(PMCID:PMC7497403)
Minard, A., Morgan, D., Raguseo, F., Di Porzio, A., Liano, D., Jamieson, A. G. and Di Antonio, M.
(2020)
A short peptide that preferentially binds c-MYC G-quadruplex DNA.
Chemical Communications, 56(63),
pp. 8940-8943.
(doi: 10.1039/D0CC02954H)
(PMID:32638724)
Magnussen, H. M. et al.
(2020)
Structural basis for DNA damage-induced phosphoregulation of MDM2 RING domain.
Nature Communications, 11,
2094.
(doi: 10.1038/s41467-020-15783-y)
(PMID:32350255)
(PMCID:PMC7190642)
Bell, J. D., Harkiss, A. H., Nobis, D., Malcolm, E., Knuhtsen, A., Wellaway, C. R., Jamieson, A. G. , Magennis, S. W. and Sutherland, A.
(2020)
Conformationally rigid pyrazoloquinazoline α-amino acids: one- and two-photon induced fluorescence.
Chemical Communications, 56(12),
pp. 1887-1890.
(doi: 10.1039/C9CC09064A)
(PMID:31956866)
Song, Y. et al.
(2020)
Mechanism of crosstalk between the LSD1 demethylase and HDAC1 deacetylase in the CoREST complex.
Cell Reports, 30(8),
2699-2711.e8.
(doi: 10.1016/j.celrep.2020.01.091)
(PMID:32101746)
2019
Alam, M. M. et al.
(2019)
Validation of the protein kinase PfCLK3 as a multistage cross-species malarial drug target.
Science, 365(6456),
eaau1682.
(doi: 10.1126/science.aau1682)
(PMID:31467193)
Mahindra, A., Millard, C. J., Black, I., Archibald, L. J., Schwabe, J. W.R. and Jamieson, A. G.
(2019)
Synthesis of HDAC substrate peptidomimetic inhibitors (SPIs) using Fmoc amino acids incorporating zinc-binding groups.
Organic Letters, 21(9),
pp. 3178-3182.
(doi: 10.1021/acs.orglett.9b00885)
(PMID:30998366)
(PMCID:PMC6503537)
Clark, G. C., Casewell, N. R., Elliott, C. T., Harvey, A. L., Jamieson, A. G. , Strong, P. N. and Turner, A. D.
(2019)
Friends or foes? Emerging impacts of biological toxins.
Trends in Biochemical Sciences, 44(4),
pp. 365-379.
(doi: 10.1016/j.tibs.2018.12.004)
(PMID:30651181)
McDougall, L. and Jamieson, A. G.
(2019)
Stapled peptides as potential therapeutics.
In:
Encyclopedia of Life Sciences.
Wiley: Chichester.
ISBN 9780470015902
(doi: 10.1002/9780470015902.a0028403)
Harkiss, A. H., Bell, J. D., Knuhtsen, A., Jamieson, A. G. and Sutherland, A.
(2019)
Synthesis and fluorescent properties of β-pyridyl α-amino acids.
Journal of Organic Chemistry, 84(5),
pp. 2879-2890.
(doi: 10.1021/acs.joc.9b00036)
(PMID:30726078)
Knuhtsen, A., Whitmore, C., McWhinnie, F. S., McDougall, L., Whiting, R., Smith, B. O. , Timperley, C. M., Green, A. C., Kinnear, K. I. and Jamieson, A. G.
(2019)
α-conotoxin GI triazole-peptidomimetics: potent and stable blockers of a human acetylcholine receptor.
Chemical Science, 10,
pp. 1671-1676.
(doi: 10.1039/C8SC04198A)
2018
Kelly, R.D.W., Chandru, A., Watson, P.J., Song, Y., Blades, M., Robertson, N.S., Jamieson, A.G. , Schwabe, J.W.R. and Cowley, S.M.
(2018)
Histone deacetylase (HDAC) 1 and 2 complexes regulate both histone acetylation and crotonylation in vivo.
Scientific Reports, 8,
14690.
(doi: 10.1038/s41598-018-32927-9)
(PMID:30279482)
(PMCID:PMC6168483)
Girt, G. C., Mahindra, A., Al Jabri, Z. J.H., De Ste Croix, M., Oggioni, M. R. and Jamieson, A. G.
(2018)
Lipopeptidomimetics derived from teixobactin have potent antibacterial activity against Staphylococcus aureus.
Chemical Communications, 54(22),
pp. 2767-2770.
(doi: 10.1039/C7CC06093A)
(PMID:29484340)
McDougall, L., Draper, E. R. , Beadle, J. D., Shipman, M., Raubo, P., Jamieson, A. G. and Adams, D.
(2018)
Enzymatically-stable oxetane-based dipeptide hydrogels.
Chemical Communications, 54(14),
pp. 1793-1796.
(doi: 10.1039/C7CC09701H)
(PMID:29384155)
2017
Beadle, J. D., Knuhtsen, A., Hoose, A., Raubo, P., Jamieson, A. G. and Shipman, M.
(2017)
Solid-phase synthesis of oxetane modified peptides.
Organic Letters, 19(12),
pp. 3303-3306.
(doi: 10.1021/acs.orglett.7b01466)
(PMID:28585839)
Pacifico, S., Kerckhoffs, A., Fallow, A. J., Foreman, R. E., Guerrini, R., McDonald, J., Lambert, D. G. and Jamieson, A. G.
(2017)
Urotensin-II peptidomimetic incorporating a non-reducible 1,5-triazole disulfide bond reveals a pseudo-irreversible covalent binding mechanism to the urotensin G-protein coupled receptor.
Organic and Biomolecular Chemistry, 15(21),
pp. 4704-4710.
(doi: 10.1039/C7OB00959C)
(PMID:28524918)
2016
Watson, P. J., Millard, C. J., Riley, A. M., Robertson, N. S., Wright, L. C., Godage, H. Y., Cowley, S. M., Jamieson, A. , Potter, B. V.L. and Schwabe, J. W.R.
(2016)
Insights into the activation mechanism of class I HDAC complexes by inositol phosphates.
Nature Communications, 7,
11262.
(doi: 10.1038/ncomms11262)
(PMID:27109927)
(PMCID:PMC4848466)
Burton, M. J. et al.
(2016)
A heme-binding domain controls regulation of ATP-dependent potassium channels.
Proceedings of the National Academy of Sciences of the United States of America, 113(14),
pp. 3785-3790.
(doi: 10.1073/pnas.1600211113)
(PMID:27006498)
(PMCID:PMC4833257)
Rennie, Y. K., McIntyre, P. J., Akindele, T., Bayliss, R. and Jamieson, A.
(2016)
A TPX2 proteomimetic has enhanced affinity for Aurora-A due to hydrocarbon stapling of a helix.
ACS Chemical Biology, 11(12),
pp. 3383-3390.
(doi: 10.1021/acschembio.6b00727)
(PMID:27775325)
2015
Jamieson, A. and Robertson, N.
(2015)
Regulation of protein–protein interactions using stapled peptides.
Reports in Organic Chemistry, 2015(5),
pp. 65-74.
(doi: 10.2147/ROC.S68161)
Hudson, G. M., Watson, P. J., Fairall, L., Jamieson, A. G. and Schwabe, J. W.R.
(2015)
Insights into the recruitment of class IIa Histone Deacetylases (HDACs) to the SMRT/NCoR transcriptional repression complex.
Journal of Biological Chemistry, 290(29),
pp. 18237-18244.
(doi: 10.1074/jbc.M115.661058)
(PMID:26055705)
(PMCID:PMC4505066)
2014
Aillard, B., Robertson, N. S., Baldwin, A. R., Robins, S. and Jamieson, A. G.
(2014)
Robust asymmetric synthesis of unnatural alkenyl amino acids for conformationally constrained α-helix peptides.
Organic and Biomolecular Chemistry, 12(43),
pp. 8775-8782.
(doi: 10.1039/C4OB01832J)
(PMID:25266495)
Evans, S. E., Goult, B. T., Fairall, L., Jamieson, A. G. , Ko Ferrigno, P., Ford, R., Schwabe, J. W.R. and Wagner, S. D.
(2014)
The ansamycin antibiotic, Rifamycin SV, inhibits BCL6 transcriptional repression and forms a complex with the BCL6-BTB/POZ domain.
PLoS ONE, 9(3),
e90889.
(doi: 10.1371/journal.pone.0090889)
(PMID:24595451)
(PMCID:PMC3942486)
2013
Jamieson, A. G. , Boutard, N., Sabatino, D. and Lubell, W. D.
(2013)
Peptide scanning for studying structure-activity relationships in drug discovery.
Chemical Biology and Drug Design, 81(1),
pp. 148-165.
(doi: 10.1111/cbdd.12042)
(PMID:23253136)
2012
Harvey, A. L., Young, L. C., Kornisiuk, E., Snitcofsky, M., Colettis, N., Blanco, C., Jerusalinsky, D., Jamieson, A. G. , Hartley, R. C. and Stone, T. W.
(2012)
A novel dihydro-pyrazolo(3,4d)(1,2,4)triazolo(1,5a)pyrimidin-4-one (AJ23) is an antagonist at adenosine A1 receptors and enhances consolidation of step-down avoidance.
Behavioural Brain Research, 234(2),
pp. 184-191.
(doi: 10.1016/j.bbr.2012.06.023)
Jamieson, A. G. , Russell, D. and Hamilton, A. D.
(2012)
A 1,3-phenyl-linked hydantoin oligomer scaffold as a β-strand mimetic.
Chemical Communications, 48(31),
pp. 3709-3711.
(doi: 10.1039/C2CC30295K)
(PMID:22399148)
2011
Adler, M. J., Jamieson, A. G. and Hamilton, A. D.
(2011)
Hydrogen-bonded synthetic mimics of protein secondary structure as disruptors of protein-protein interactions.
In: Vassilev, L. and Fry, D. (eds.)
Small-Molecule Inhibitors of Protein-Protein Interactions.
Series: Current topics in microbiology and immunology, 348 (348).
Springer, pp. 1-23.
ISBN 9783642170829
(doi: 10.1007/82_2010_91)
2010
Ronga, L., Jamieson, A. G. , Beauregard, K., Quiniou, C., Chemtob, S. and Lubell, W. D.
(2010)
Insertion of multiple α-amino γ-lactam (Agl) residues into a peptide sequence by solid-phase synthesis on synphase lanterns.
Biopolymers, 94(2),
pp. 183-191.
(doi: 10.1002/bip.21288)
Boutard, N., Jamieson, A. G. , Ong, H. and Lubell, W. D.
(2010)
Structure-activity analysis of the growth hormone Secretagogue GHRP-6 by α- and β-amino γ-lactam positional scanning.
Chemical Biology and Drug Design, 75(1),
pp. 40-50.
(doi: 10.1111/j.1747-0285.2009.00913.x)
St-Cyr, D. J., Jamieson, A. G. and Lubell, W. D.
(2010)
α-Amino-β-hydroxy-γ-lactam for constraining peptide Ser and Thr residue conformation.
Organic Letters, 12(8),
pp. 1652-1655.
(doi: 10.1021/ol1000582)
2009
Bourguet, C. B. et al.
(2009)
Portraits of the pioneers of the American Peptide Society.
In: Del Valle, S., Escher, E. and Lubell, W. D. (eds.)
Peptides for Youth.
Series: Advances in experimental medicine and biology (611).
Springer, xlix-lxix.
ISBN 9780387736563
Jamieson, A. G. , Boutard, N., Beauregard, K., Bodas, M. S., Ong, H., Quiniou, C., Chemtob, S. and Lubell, W. D.
(2009)
Positional scanning for peptide secondary structure by systematic solid-phase synthesis of amino lactam peptides.
Journal of the American Chemical Society, 131(22),
pp. 7917-7927.
(doi: 10.1021/ja9010628)
(PMID:19453183)
2007
Jamieson, A. G. and Sutherland, A.
(2007)
Ether-directed palladium(II)-catalysed aza-Claisen rearrangements: studies on the origin of the directing effect.
Tetrahedron, 63,
pp. 2123-2131.
(doi: 10.1016/j.tet.2006.12.067)
Jamieson, A. G. and Sutherland, A.
(2007)
Ether-directed, stereoselective aza-Claisen rearrangements: Synthesis of the piperidine alkaloid, alpha-conhydrine.
Organic Letters, 9,
pp. 1609-1611.
(doi: 10.1021/ol070424z)
(PMID:17371038)
2006
Fanning, K. N., Jamieson, A. G. and Sutherland, A.
(2006)
Palladium(II)-catalysed rearrangement reactions.
Current Organic Chemistry, 10(9),
pp. 1007-1020.
(doi: 10.2174/138527206777435490)
Jamieson, A. G. and Sutherland, A.
(2006)
Scope and limitations of ether-directed, metal-catalysed aza-Claisen rearrangements; improved stereoselectivity using non-coordinating solvents.
Organic and Biomolecular Chemistry, 4,
pp. 2932-2937.
(doi: 10.1039/b607014k)
(PMID:16855742)
2005
Fanning, K. N., Jamieson, A. G. and Sutherland, A.
(2005)
Stereoselective beta-hydroxy-alpha-amino acid synthesis via an ether-directed, palladium-catalysed aza-Claisen rearrangement.
Organic and Biomolecular Chemistry, 3,
pp. 3749-3756.
(doi: 10.1039/b510808j)
(PMID:16211111)
Jamieson, A. G. and Sutherland, A.
(2005)
A highly stereoselective ether directed palladium catalysed aza-Claisen rearrangement.
Organic and Biomolecular Chemistry, 3,
pp. 735-736.
(PMID:15731857)
2004
Jamieson, A. G. , Sutherland, A. and Willis, C. L.
(2004)
The first enantioselective synthesis of the amino acid, (2S,3S,4R)-gamma-hydroxyisoleucine using a palladium(II) catalysed 3,3-sigmatropic rearrangement.
Organic and Biomolecular Chemistry, 2,
pp. 808-809.
(doi: 10.1039/b401076k)
This list was generated on Wed Jun 7 15:51:58 2023 BST.